Tarlatamab

Tarlatamab
Monoclonal antibody
TypeBi-specific T-cell engager
SourceHuman
TargetDLL3 and CD3
Clinical data
Trade namesImdelltra
Other namesAMG757; AMG-757, tarlatamab-dlle
AHFS/Drugs.comMultum Consumer Information
License data
Routes of
administration
Intravenous
Drug classAntineoplastic
ATC code
Legal status
Legal status
Identifiers
CAS Number
DrugBank
UNII
KEGG
Chemical and physical data
FormulaC4664H7139N1259O1454S34
Molar mass105202.82 g·mol−1

Tarlatamab, sold under the brand name Imdelltra, is an anti-cancer medication used for the treatment of extensive-stage small cell lung cancer. It is a bispecific T-cell engager that binds delta-like ligand 3 and CD3.

The most common adverse reactions include cytokine release syndrome, fatigue, pyrexia, dysgeusia, decreased appetite, musculoskeletal pain, and constipation, anemia and nausea.

Tarlatamab was approved for medical use in the United States in May 2024. The US Food and Drug Administration (FDA) considers it to be a first-in-class medication.