Eptazocine

Eptazocine
Clinical data
Routes of; administration	Oral
ATC code	None;
Legal status
Legal status	In general: ℞ (Prescription only);
Identifiers
	IUPAC name (1S,6S)-1,4-dimethyl-2,3,4,5,6,7-hexahydro-1H-1,6-methano-4-benzazonin-10-ol;
CAS Number	72522-13-5 ; 72150-17-5 (bromide);
PubChem CID	3042090;
ChemSpider	2305268;
UNII	2208ZLI77S;
ChEMBL	ChEMBL70566;
CompTox Dashboard (EPA)	DTXSID501024513 ;
Chemical and physical data
Formula	C15H21NO
Molar mass	231.339 g·mol−1
3D model (JSmol)	Interactive image;
	SMILES Oc1ccc2c(c1)[C@@]3(CCN(C[C@H](C2)C3)C)C;
	InChI InChI=1S/C15H21NO/c1-15-5-6-16(2)10-11(9-15)7-12-3-4-13(17)8-14(12)15/h3-4,8,11,17H,5-7,9-10H2,1-2H3/t11-,15-/m1/s1; Key:ZOWQTJXNFTWSCS-IAQYHMDHSA-N;

Eptazocine (Sedapain) is an opioid analgesic which was introduced in Japan by Morishita in 1987. It acts as a mixed κ-opioid receptor agonist and μ-opioid receptor antagonist.

Clinical data


Routes of administration	Oral
ATC code	None
Legal status
Legal status	In general: ℞ (Prescription only)
Identifiers
IUPAC name (1S,6S)-1,4-dimethyl-2,3,4,5,6,7-hexahydro-1H-1,6-methano-4-benzazonin-10-ol
CAS Number	72522-13-5 72150-17-5 (bromide)
PubChem CID	3042090
ChemSpider	2305268
UNII	2208ZLI77S
ChEMBL	ChEMBL70566
CompTox Dashboard (EPA)	DTXSID501024513
Chemical and physical data
Formula	C₁₅H₂₁NO
Molar mass	231.339 g·mol⁻¹
3D model (JSmol)	Interactive image
SMILES Oc1ccc2c(c1)[C@@]3(CCN(C[C@H](C2)C3)C)C
InChI InChI=1S/C15H21NO/c1-15-5-6-16(2)10-11(9-15)7-12-3-4-13(17)8-14(12)15/h3-4,8,11,17H,5-7,9-10H2,1-2H3/t11-,15-/m1/s1 Key:ZOWQTJXNFTWSCS-IAQYHMDHSA-N